Piero Temperini

Piero Temperini

PhD fellow


Publication year:
  1. 2019
  2. Published

    N-(7-(1H-imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide - a new kainate receptor selective antagonist and analgesic: Synthesis, X-ray crystallography, structure-affinity relationships, in vitro and in vivo pharmacology

    Møllerud, S., Hansen, R. B., Pallesen, J. S., Temperini, Piero, Pasini, D., Bornholdt, J., Nielsen, Birgitte, Mamedova, Esmira, Chalupnik, P., Paternain, A. V., Lerma, J., Del Castillo, M. D., Andreasen T., Jesper, Frydenvang, Karla Andrea, Kastrup, Jette Sandholm Jensen, Johansen, Tommy Nørskov & Pickering, Darryl S, 2019, In: ACS Chemical Neuroscience. 10, p. 4685-4695 11 p.

    Research output: Contribution to journalJournal articlepeer-review

  3. 2020
  4. Published

    Stereoselective Synthesis of New (2S,3R)-3-Carboxyphenyl)pyrrolidine-2-carboxylic Acid Analogues Utilizing a C(sp3)-H Activation Strategy and Structure-Activity Relationship Studies at the Ionotropic Glutamate Receptors

    Kayser, S., Hansen, J. C., Staudt, Markus, Moroz, A., Larsen, Y., Temperini, Piero, Yi, F., Syrenne, J. T., Krogsgaard-Larsen, N., Iliadis, S., Nielsen, Birgitte, Hansen, K. B., Pickering, Darryl S & Bunch, Lennart, 2020, In: ACS Chemical Neuroscience. 11, p. 674-701 28 p.

    Research output: Contribution to journalJournal articlepeer-review

  5. Published
  6. 2021
  7. Published

    Structure of the mini-RNA-guided endonuclease CRISPR-Cas12j3

    Carabias del Rey, Arturo, Fuglsang, Anders, Temperini, Piero, Pape, T., Sofos, N., Stella, S., Erlendsson, Simon & Montoya, Guillermo, 2021, In: Nature Communications. 12, 12 p., 4476.

    Research output: Contribution to journalJournal articlepeer-review

  8. 2024
  9. Accepted/In press

    Tritium and deuterium labelling of a kainate receptor antagonist and evaluation as a radioligand

    Chałupnik, P., Marek, A., Hovah, M. E. L., Pickering, Darryl S, Temperini, Piero, Donbosco, S., Szymańska, E. & Johansen, Tommy Nørskov, 2024, (Accepted/In press) In: Journal of Labelled Compounds and Radiopharmaceuticals.

    Research output: Contribution to journalJournal articlepeer-review

ID: 230329841